Auflistung Universitätsbibliographie nach Autor "Kudolo, Mark"

Anzeige der Dokumente 1-17 von 17

Bioisosteric Replacement of Arylamide-Linked Spine Residues with N-Acylhydrazones and Selenophenes as a Design Strategy to Novel Dibenzosuberone Derivatives as Type I 1/2 p38 alpha MAP Kinase Inhibitors

Pedreira, Julia G. B.; Nahidino, Philipp; Kudolo, Mark; Pantsar, Tatu; Berger, Benedict-Tilman; Forster, Michael; Knapp, Stefan; Laufer, Stefan; Barreiro, Eliezer J. (2020)
Decisive role of water and protein dynamics in residence time of p38 alpha MAP kinase inhibitors

Pantsar, Tatu; Kaiser, Philipp D.; Kudolo, Mark; Forster, Michael; Rothbauer, Ulrich; Laufer, Stefan A. (2022)
Design, Synthesis and Biological Evaluation of 7-Chloro-9H-pyrimido[4,5-b]indole-based Glycogen Synthase Kinase-3 beta Inhibitors

Andreev, Stanislav; Pantsar, Tatu; Ansideri, Francesco; Kudolo, Mark; Forster, Michael; Schollmeyer, Dieter; Laufer, Stefan A.; Koch, Pierre (2019)
Development of a Selective Dual Discoidin Domain Receptor (DDR)/p38 Kinase Chemical Probe

Roehm, Sandra; Berger, Benedict-Tilman; Schroeder, Martin; Chatterjee, Deep; Mathea, Sebastian; Joerger, Andreas C.; Pinkas, Daniel M.; Bufton, Joshua C.; Tjaden, Amelie; Kovooru, Lohitesh; Kudolo, Mark; Pohl, Christian; Bullock, Alex N.; Mueller, Susanne; Laufer, Stefan; Knapp, Stefan (2021)
Development of novel urea-based ATM kinase inhibitors with subnanomolar cellular potency and high kinome selectivity

Dimitrov, Teodor; Anli, Cetin; Moschopoulou, Athina Anastasia; Kronenberger, Thales; Kudolo, Mark; Geibel, Christian; Schwalm, Martin Peter; Knapp, Stefan; Zender, Lars; Forster, Michael; Laufer, Stefan (2022)
Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor

Serafim, Ricardo A. M.; Santiago, Andre da Silva; Schwalm, Martin P.; Hu, Zexi; dos Reis, Caio, V; Takarada, Jessica E.; Mezzomo, Priscila; Massirer, Katlin B.; Kudolo, Mark; Gerstenecker, Stefan; Chaikuad, Apirat; Zender, Lars; Knapp, Stefan; Laufer, Stefan; Counago, Rafael M.; Gehringer, Matthias (2022)
Discovery and Development of First-in-Class ACKR3/CXCR7 Superagonists for Platelet Degranulation Modulation

Bayrak, Alp; Mohr, Florian; Kolb, Kyra; Szpakowska, Martyna; Shevchenko, Ekaterina; Dicenta, Valerie; Rohlfing, Anne-Katrin; Kudolo, Mark; Pantsar, Tatu; Guenther, Marcel; Kaczor, Agnieszka A.; Poso, Antti; Chevigne, Andy; Pillaiyar, Thanigaimalai; Gawaz, Meinrad; Laufer, Stefan A. (2022)
Discovery and Evaluation of Enantiopure 9H-pyrimido[4,5-b]indoles as Nanomolar GSK-3 beta Inhibitors with Improved Metabolic Stability

Andreev, Stanislav; Pantsar, Tatu; El-Gokha, Ahmed; Ansideri, Francesco; Kudolo, Mark; Anton, Debora Bublitz; Sita, Giulia; Romasco, Jenny; Geibel, Christian; Laemmerhofer, Michael; Goettert, Marcia Ines; Tarozzi, Andrea; Laufer, Stefan A.; Koch, Pierre (2020)
Discovery of a Potent and Highly Isoform-Selective Inhibitor of the Neglected Ribosomal Protein S6 Kinase Beta 2 (S6K2)

Gerstenecker, Stefan; Haarer, Lisa; Schroder, Martin; Kudolo, Mark; Schwalm, Martin P.; Wydra, Valentin; Serafim, Ricardo A. M.; Chaikuad, Apirat; Knapp, Stefan; Laufer, Stefan; Gehringer, Matthias (2021)
Discovery of potent p38 alpha MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation

Astolfi, Andrea; Kudolo, Mark; Brea, Jose; Manni, Giorgia; Manfroni, Giuseppe; Palazzotti, Deborah; Sabatini, Stefano; Cecchetti, Federica; Felicetti, Tommaso; Cannalire, Rolando; Massari, Serena; Tabarrini, Oriana; Loza, Maria Isabel; Fallarino, Francesca; Cecchetti, Violetta; Laufer, Stefan A.; Barreca, Maria Letizia (2019)
Fast Iterative Synthetic Approach toward Identification of Novel Highly Selective p38 MAP Kinase Inhibitors

Roehm, Sandra; Berger, Benedict-Tilman; Schroeder, Martin; Chaikuad, Apirat; Winkel, Rob; Hekking, Koen F. W.; Benningshof, Jorg J. C.; Mueller, Gerhard; Tesch, Roberta; Kudolo, Mark; Forster, Michael; Laufer, Stefan; Knapp, Stefan (2019)
From 2-Alkylsulfanylimidazoles to 2-Alkylimidazoles: An Approach towards Metabolically More Stable p38 alpha MAP Kinase Inhibitors

Heider, Fabian; Haun, Urs; Doering, Eva; Kudolo, Mark; Sessler, Catharina; Albrecht, Wolfgang; Laufer, Stefan; Koch, Pierre (2017)
Gefitinib-Tamoxifen Hybrid Ligands as Potent Agents against Triple-Negative Breast Cancer

Abdelmalek, Carine M.; Hu, Zexi; Kronenberger, Thales; Kublbeck, Jenni; Kinnen, Franziska J. M.; Hesse, Salma S.; Malik, Afsin; Kudolo, Mark; Niess, Raimund; Gehringer, Matthias; Zender, Lars; Witt-Enderby, Paula A.; Zlotos, Darius P.; Laufer, Stefan A. (2022)
Pyridinylimidazoles as dual glycogen synthase kinase 3 beta/p38 alpha mitogen-activated protein kinase inhibitors

Heider, Fabian; Ansideri, Francesco; Tesch, Roberta; Pantsar, Tatu; Haun, Urs; Doering, Eva; Kudolo, Mark; Poso, Antti; Albrecht, Wolfgang; Laufer, Stefan A.; Koch, Pierre (2019)
Pyridinylimidazoles as GSK3 beta Inhibitors: The Impact of Tautomerism on Compound Activity via Water Networks

Heider, Fabian; Pantsar, Tatu; Kudolo, Mark; Ansideri, Francesco; De Simone, Angela; Pruccoli, Letizia; Schneider, Taiane; Goettert, Marcia Ines; Tarozzi, Andrea; Andrisano, Vincenza; Laufer, Stefan A.; Koch, Pierre (2019)
Selective targeting of the alpha C and DFG-out pocket in p38 MAPK

Roehm, Sandra; Schroeder, Martin; Dwyer, Jessica E.; Widdowson, Caroline S.; Chaikuad, Apirat; Berger, Benedict-Tilman; Joerger, Andreas C.; Kraemer, Andreas; Harbig, Jule; Dauch, Daniel; Kudolo, Mark; Laufer, Stefan; Bagley, Mark C.; Knapp, Stefan (2020)
Structural Optimization of a Pyridinylimidazole Scaffold: Shifting the Selectivity from p38 alpha Mitogen-Activated Protein Kinase to c-Jun N-Terminal Kinase 3

Ansideri, Francesco; Macedo, Joana T.; Eitel, Michael; El-Gokha, Ahmed; Zinad, Dhafer S.; Scarpellini, Camilla; Kudolo, Mark; Schollmeyer, Dieter; Boeckler, Frank M.; Blaum, Baerbel S.; Laufer, Stefan A.; Koch, Pierre (2018)

Anzeige der Dokumente 1-17 von 17

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Auflistung Universitätsbibliographie nach Autor "Kudolo, Mark"

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